Azatadine Maleate ( Azatadine Maleate; azatadine; azatadine maleate; Idulamine; Idulian )

产品货号. M14367 CAS No. 3978-86-7

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

Azatadine Maleate
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

Azatadine dimaleate is an histamine and cholinergic inhibitor with IC50 of 6.5 nM and 10 nM, respectively.
产品描述

Azatadine dimaleate is an histamine and cholinergic inhibitor with IC50 of 6.5 nM and 10 nM, respectively.
同义词

Azatadine Maleate; azatadine; azatadine maleate; Idulamine; Idulian
通路

Endocrinology/Hormones
靶点

5-HT Receptor
受体

HT; Cholinergic
研究领域

Inflammation/Immunology
适应症

——

CAS Number

3978-86-7
分子量

522.55
分子式

C28H30N2O8
纯度

>98%(HPLC)
溶解度

Water: 105 mg/mL (200.93 mM); DMSO: 105 mg/mL (200.93 mM)
SMILES

CN1CC/C(CC1)=C2C3=CC=CC=C3CCC4=CC=CN=C4\2.O=C(O)/C=C\C(O)=O.O=C(O)/C=C\C(O)=O
化学全称

6,11-Dihydro-11-(1-methylpiperidin-4-ylidene)-5H-benzo[5,6]cyclohepta[1,2-b]pyridine dimaleate

1.Tozzi S, et al. Agents Actions, 1974, 4(4), 264-270.

计算器

产品手册

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